- norethisterone. The
progestins are
structural analogues of
progesterone and have
progestogenic activity similarly, but
differ from
progesterone in
their pharmacological...
-
etonogestrel (3-ketodesogestrel), and, via this
active metabolite, it has
progestogenic activity,
antigonadotropic effects, very weak
androgenic activity, very...
-
strong anabolic effects and
highly androgenic effects, as well as
potent progestogenic effects, and weak
glucocorticoid effects.
Trenbolone acetate is an androgen...
-
among others.
Tibolone is a
synthetic steroid with weak estrogenic,
progestogenic, and
androgenic activity, and
hence is an
agonist of the estrogen, progesterone...
- has
progestogenic and
antimineralocorticoid activity. The loss of the C7α
acetylthio group of spironolactone, a
compound with
negligible progestogenic activity...
-
target of
progestogens like progesterone. Due to its
androgenic and
progestogenic activity,
trestolone has
antigonadotropic effects.
These effects result...
-
bioavailability and
metabolic stability with
dydrogesterone as well as
additional progestogenic activity of its metabolites.
Dydrogesterone binds to and
activates both...
-
replacement dosages (0.35 to 1 mg/day),
norethisterone has
essentially progestogenic side
effects only. In most
clinical studies of
norethisterone for contraception...
- the
progesterone and
estrogen receptors and to have very weak
mixed progestogenic and
antiprogestogenic activity as well as very weak
mixed estrogenic...
-
Progestogens are
agonists of the
progesterone receptors (PRs) and
produce progestogenic, or progestational, effects. They have
important effects in the female...
