- Antiestrogens, also
known as
estrogen antagonists or
estrogen blockers, are a
class of
drugs which prevent estrogens like
estradiol from
mediating their...
- IA and
their balance of
estrogenic and
antiestrogenic activity.
Raloxifene is a SERM that is more
antiestrogenic than tamoxifen; both are
estrogenic in...
- Anastrozole, sold
under the
brand name
Arimidex among others, is an
antiestrogenic medication used in
addition to
other treatments for
breast cancer. Specifically...
- 4-hydroxyestrone all are. In addition,
although not
antiestrogenic in the uterus, 2-hydroxyestrone
shows antiestrogenic effects on
luteinizing hormone and prolactin...
-
estrogenic and
antiestrogenic activity, with its
profile of
effects differing by tissue. For instance,
tamoxifen has
predominantly antiestrogenic effects in...
- of the
estrogen receptor (ER). It has
estrogenic effects in bone and
antiestrogenic effects in the **** and uterus.
Raloxifene was
approved for medical...
-
breast cancer. The drug is
described as
slightly estrogenic and
potently antiestrogenic, and
inhibits mammary gland development and
suppresses prolactin levels...
- lunamarine,
isolated from B.
diffusa has
shown some in
vitro anticancer,
antiestrogenic, immunomodulatory, and anti-amoebic
activity (particularly
against Entamoeba...
-
estrogen levels. Conversely, it is an
antagonist of the ERĪ².
Clomifene has
antiestrogenic effects in the uterus.
There is
little clinical research on the influence...
-
Because of its
progestogenic activity,
progesterone has
functional antiestrogenic effects in
certain tissues such as the uterus, cervix, and ****. In...
