-
analogues (both
agonists and antagonists). However, many
other drugs have
antigonadotropic properties as well,
including compounds acting on ****
steroid hormone...
- glucocorticoid, or
antimineralocorticoid activity. They also have
antigonadotropic effects and at high
doses can
strongly suppress ****
hormone production...
- off-target
activity in the
antiandrogen in question. For instance,
whereas antigonadotropic antiandrogens like GnRH
modulators and
cyproterone acetate are ****ociated...
- (3-ketodesogestrel), and, via this
active metabolite, it has
progestogenic activity,
antigonadotropic effects, very weak
androgenic activity, very weak
glucocorticoid activity...
- 6 mg per cycle. Due to its
progestogenic activity,
levonorgestrel has
antigonadotropic effects and is able to
suppress the
secretion of the gonadotropins...
-
menstrual bleeding relative to
progestogen exposure alone. NETA has
antigonadotropic effects via its
progestogenic activity and can dose-dependently suppress...
- activity. Due to its
progestogenic activity,
megestrol acetate has
antigonadotropic effects. The
mechanism of
action of the
appetite stimulant effects...
-
activation of the PR and AR in the
pituitary gland,
danazol produces antigonadotropic effects.
Although its does not
significantly affect basal luteinizing...
-
membrane estrogen receptor,
similarly to estradiol.
Estrogens have
antigonadotropic effects through activation of the ERα. As a contraceptive, ethinylestradiol...
- been
described as "special" progestogen,
possessing low or
moderate antigonadotropic efficacy but
strong or very
strong endometrial efficacy. In relation...
