-
Ethisterone, also
known as ethinyltestosterone, pregneninolone, and
anhydrohydroxyprogesterone and
formerly sold
under the
brand names Proluton C and...
- 17α-Ethynylated/vinylated
testosterone derivatives:
ethynyltestosterone (
ethisterone) and
vinyltestosterone derivatives The last
group consists of progestins...
-
derived from
modification of
ethisterone via
introduction of
methyl groups at the C6α and C21 positions.
Relative to
ethisterone, it is 12 times as potent...
-
affinity and
efficacy of
danazol itself at the PR are
relatively low,
ethisterone, one of the
major metabolites of danazol, is
described as a weak progestogen...
- to
ethisterone and
shows about half its
progestogenic potency.
Ethinylandrostenediol was an
intermediate in the
initial synthesis of
ethisterone. Ethinylandrostenediol...
-
usually administered doses is the
androgen danazol, a
derivative of
ethisterone (ethinyltestosterone).
Fetal masculinization of the **** has resulted...
-
metabolite of the
formerly clinically used but now-discontinued
progestin ethisterone and the
experimental and never-marketed
hormonal antineoplastic agent...
- Also
sometimes designed as
ethinyl in
compounds (ethinylestradiol,
ethisterone (ethinyltestosterone)). See main page alkynes.
Ethynyl radical (HC≡C·)...
- was
first introduced for
medical use in 1934 and the
first progestin,
ethisterone, was
introduced for
medical use in 1939. More
potent progestins, such...
-
group greatly reduces but does not
abolish androgenic activity, as in
ethisterone (17α-ethynyltestosterone) and
norethisterone (17α-ethynyl-19-nortestosterone)...
