-
Astemizole (marketed
under the
brand name Hismanal,
developmental code R43512) was a second-generation
antihistamine drug that has a long
duration of action...
-
Xenopus oocytes by the
histamine receptor antagonists terfenadine and
astemizole". FEBS Letters. 385 (1–2): 77–80. doi:10.1016/0014-5793(96)00355-9. PMID 8641472...
- QT interval.
Other examples include terfenadine (Seldane, Seldane-D),
astemizole (Hismanal),
cisapride (Propulsid,
withdrawn in many
countries for prolonging...
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selectively binding and
depolymerising their tubulins.
Antihistamines such as
astemizole, bilastine, clemizole, emedastine, mizolastine, and oxatomide. Benzimidazole...
-
delavirdine fluvoxamine iron
salts voriconazole aminophylline and
theophylline astemizole It is a
racemic 1:1
mixture of the
enantiomers dexlansoprazole and levolansoprazole...
-
causing prolonged QT
interval (on EKG) or wave-burst
arrhythmia (i.e.:
astemizole, bepridil, IV erythromycin, halofantrine, pentamidine, sultopride, terfenadine...
- In some cases, this can lead to a
fatal interaction with
drugs like
astemizole or terfenadine. The
effect of
grapefruit juice with
regard to drug absorption...
-
antihistamines include:
Acrivastine (Benadryl
Allergy Relief (UK), Semprex-D (US))
Astemizole (Hismanal) –
withdrawn Bepotastine (Talion, Bepreve)
Bilastine (Blexten...
-
histamine H1-receptors (Ki=64 nM) with an
affinity comparable to that of
astemizole and diphenhydramine, and
superior than that of
cetirizine by three-fold...
- of
clarithromycin with the
following medications: cisapride, pimozide,
astemizole, terfenadine, ergotamine, ticagrelor,
ranolazine or dihydroergotamine...
