- concentration) 50–72 (EC50Tooltip Half-maximal
effective concentration) (rat)
NETTooltip Norepinephrine transporter 27,000–30,500 (Ki) 360–405 (IC50) 54–110 (EC50)...
- MK-801/PCPTooltip
phencyclidine site
SERTTooltip Serotonin transporter and
NETTooltip norepinephrine transporter blocker (cf. serotonin–norepinephrine reuptake...
- Site CBP NCBP
Action SERTTooltip Serotonin transporter 108 ND
Inhibitor NETTooltip Norepinephrine transporter 36 ND
Inhibitor DATTooltip Dopamine transporter...
- (SERTTooltip
serotonin transporter,
DATTooltip dopamine transporter,
NETTooltip norepinephrine transporter). It is ****ociated with
monoamine reuptake...
- 000 (Ki) >100,000 (IC50Tooltip half-maximal
inhibitory concentration)
NETTooltip Norepinephrine transporter 5,600–>30,000 (Ki) >100,000 (IC50) DATTooltip...
-
DATTooltip Dopamine transporter (DRIsTooltip
Dopamine reuptake inhibitors)
NETTooltip Norepinephrine transporter (NRIsTooltip
Norepinephrine reuptake inhibitors)...
-
Partial Agonist Rat
SERTTooltip Serotonin transporter 2,234
Inhibitor Human NETTooltip Norepinephrine transporter >10,000
Inhibitor Human DATTooltip Dopamine...
- receptor, or the
monoamine transporters (SERTTooltip
serotonin transporter,
NETTooltip norepinephrine transporter, or
DATTooltip dopamine transporter) at the...
- Site ATX 4-OH-ATX N-DM-ATX
SERTTooltip Serotonin transporter 77 43 ND
NETTooltip Norepinephrine transporter 5 3 92 DAT 1,451 ND ND
MORTooltip μ-Opioid...
- (HNK) IC50 NAM Rat ERαTooltip
Estrogen receptor alpha 0.34 Ki ND
Human NETTooltip Norepinephrine transporter 82–291 IC50
Inhibitor Human DATTooltip Dopamine...