- (SERTTooltip
serotonin transporter,
NETTooltip norepinephrine transporter, or
DATTooltip dopamine transporter) at the ****essed
concentrations (Ki = >7,510–10,550 nM)...
-
Norepinephrine transporter 27,000–30,500 (Ki) 360–405 (IC50) 54–110 (EC50) (rat)
DATTooltip Dopamine transporter 6,500–>10,000 (Ki) 1,440–21,000 (IC50) 51–278 (EC50)...
-
sites on the
monoamine transporters (SERTTooltip
serotonin transporter,
DATTooltip dopamine transporter,
NETTooltip norepinephrine transporter). It is ****ociated...
- 108 ND
Inhibitor NETTooltip Norepinephrine transporter 36 ND
Inhibitor DATTooltip Dopamine transporter 5489 ND
Inhibitor 5-HT1A 5300 3200
Agonist 5-HT2A...
-
NETTooltip Norepinephrine transporter 5,600–>30,000 (Ki) >100,000 (IC50)
DATTooltip Dopamine transporter >30,000 (Ki) >100,000 (IC50) Notes: The
smaller the...
-
Norepinephrine transporter 6,500–>10,000 (Ki) 3,900 (IC50) 4,166 (EC50)
DATTooltip Dopamine transporter >10,000–22,000 (Ki) 52,000 (IC50) >10,000 (EC50)...
- 23–40 401–484 Rat
NETTooltip Norepinephrine transporter 240+ 340+ Rat
DATTooltip Dopamine transporter 1000+ 1000+ Rat 5-HT1A 1000+ 1000+ Rat 5-HT1B/1D...
-
Human NETTooltip Norepinephrine transporter 82–291 IC50
Inhibitor Human DATTooltip Dopamine transporter 63 Ki
Inhibitor Rat HCN1Tooltip Hyperpolarization-activated...
-
NETTooltip Norepinephrine transporter 13,000 (Ki) 14,000 (IC50) >10,000 (EC50)
DATTooltip Dopamine transporter 6,000–>30,000 (Ki) >100,000 (IC50) >10,000 (EC50)...
- v t e
Monoamine reuptake inhibitors DATTooltip Dopamine transporter (DRIsTooltip
Dopamine reuptake inhibitors)
NETTooltip Norepinephrine transporter (NRIsTooltip...
