-
Enkephalinases are
enzymes that
degrade endogenous enkephalin opioid peptides. They include:
Aminopeptidase N (APN)
Neutral endopeptidase (NEP) Dipeptidyl...
- An
enkephalinase inhibitor is a type of
enzyme inhibitor which inhibits one or more
members of the
enkephalinase class of
enzymes that
break down the...
- acetorphan, is an
antidiarrheal medication which acts as a
peripheral enkephalinase inhibitor.
Unlike other opioid medications used to
treat diarrhea, which...
-
identical to
somatostatin receptors (SSTRs).[citation needed]
Endorphin Enkephalinase Opioid peptide Racecadotril RB-101 PDB: 1plx;
Marcotte I, Separovic...
- an
enkephalinase inhibitor.
Spillantini MG,
Geppetti P,
Fanciullacci M,
Michelacci S,
Lecomte JM,
Sicuteri F (June 1986). "In vivo '
enkephalinase' inhibition...
-
Opioid modulator Opioid receptor agonist Opioid receptor antagonist Enkephalinase inhibitor Other Adenosine reuptake inhibitor (AdoRI)
Angiotensin II...
- also
comprise allosteric modulators and
enzyme affecting agents like
enkephalinase inhibitors. BMS-986121: μ-PAM BMS-986122: μ-PAM
Ignavine Oxytocin: μ-PAM...
- M, et al. (2000). "Thiorphan, an
inhibitor of
neutral endopeptidase/
enkephalinase (CD10/CALLA)
enhances cell
proliferation in bone
marrow cultures of...
-
analogue of RB-101. It acts as an
enkephalinase inhibitor,
which is used in
scientific research. RB-101 -
enkephalinase inhibitor that
produces analgesia...
- μ-opioid (MOR) δ-opioid (DOR) κ-opioid (KOR)
Nociceptin (NOP)
Others Enkephalinase inhibitors:
Amastatin BL-2401
Candoxatril D -Phenylalanine Dexecadotril...
