-
Enkephalinases are
enzymes that
degrade endogenous enkephalin opioid peptides. They include:
Aminopeptidase N (APN)
Neutral endopeptidase (NEP) Dipeptidyl...
- An
enkephalinase inhibitor is a type of
enzyme inhibitor which inhibits one or more
members of the
enkephalinase class of
enzymes that
break down the...
- acetorphan, is an
antidiarrheal medication which acts as a
peripheral enkephalinase inhibitor.
Unlike other opioid medications used to
treat diarrhea, which...
- 2000s. D-Phenylalanine has been
found to act as an
enkephalinase inhibitor, an
inhibitor of
enkephalinase enzymes that
break down
endogenous opioid peptides...
- unknown. It
might interact with
certain melanocortin receptors or
inhibit enkephalinase enzymes. Chemically,
Semax is a
peptide and a
synthetic analogue of...
-
disorder D-Phenylalanine (DPA, D-Phe; Deprenon, Sabiben, Sabiden) –
enkephalinase inhibitor Agomelatine (Valdoxan) – 5-HT2C
receptor antagonist and MT1...
-
identical to
somatostatin receptors (SSTRs).[citation needed]
Endorphin Enkephalinase Opioid peptide Racecadotril RB-101 PDB: 1plx;
Marcotte I, Separovic...
- μ-opioid (MOR) δ-opioid (DOR) κ-opioid (KOR)
Nociceptin (NOP)
Others Enkephalinase inhibitors:
Amastatin BL-2401
Candoxatril D-Phenylalanine Dexecadotril...
- an
enkephalinase inhibitor.
Spillantini MG,
Geppetti P,
Fanciullacci M,
Michelacci S,
Lecomte JM,
Sicuteri F (June 1986). "In vivo '
enkephalinase' inhibition...
-
acting at δ- and μ-opioid receptors, and so can also be
produced by
enkephalinase inhibitors such as RB-101. However, in
human models the data for antidepressant...
