-
Toremifene, sold
under the
brand name
Fareston among others, is a
medication which is used in the
treatment of
advanced breast cancer in postmenopausal...
- hot flushes.
Ospemifene is an
analogous metabolite of
toremifene.
Unlike tamoxifen,
toremifene is not a rat
hepatocarcinogen and
therefore ospemifene...
- in 2001, and
reincorporated in
Delaware in 2003. The
company licensed toremifene from
Orion Corporation, and
licensed andarine,
enobosarm and prostarine...
-
Raloxifene Rimostil (P-081)
Spironolactone SS1010
Tamoxifen TAS-108 (SR-16234)
Toremifene Trioxifene TZE-5323 U-11555A U-11634 Y-134
Zindoxifene Zuclomifene Antagonists...
- deaminohydroxytoremifene),
raloxifene (Evista),
tamoxifen (Nolvadex), and
toremifene (Fareston; 4-chlorotamoxifen).
SERMs that are
currently under development...
-
postmenopausal women.
Toremifene is a
similar SERM drug to tamoxifen, but is less
common and only
approved for
treatment of
metastatic cancer.
Toremifene is generally...
- 4-Hydroxytamoxifen; 4-OHT 100.1 (1.7–257) 10 (0.98–339) 2.3 (0.1–3.61) 0.04–4.8 SERM
Toremifene 4-Chlorotamoxifen; 4-CT ? ? 7.14–20.3 15.4 SERM
Clomifene MRL-41 25 (19...
-
Selective estrogen receptor modulators,
including raloxifene,
tamoxifen and
toremifene are banned. Clomiphene, cyclofenil, fulvestrant, and all
other anti-estrogenic...
- miproxifene,
miproxifene phosphate, nafoxidine, ospemifene, panomifene, and
toremifene. The
antiestrogen ethamoxytriphetol (MER-25) is also
closely related,...
-
Raloxifene Rimostil (P-081)
Spironolactone SS1010
Tamoxifen TAS-108 (SR-16234)
Toremifene Trioxifene TZE-5323 U-11555A U-11634 Y-134
Zindoxifene Zuclomifene Antagonists...