-
Funapide (INN;
former developmental codes TV-45070 and XEN402) is a
novel analgesic under development by
Xenon Pharmaceuticals (formerly in partnership...
- Nav1.7 and Nav1.8 voltage-gated
sodium channels, such as CNV1014802 and
Funapide, are
being investigated as
novel analgesics.
Sodium channel opener...
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mirogabalin and pregabalin),
activated sodium channel (VGSC)
blockade (
funapide and lidocaine), cyclooxygenase-1 (COX-1)
inhibition (TRK-700), adapter-****ociated...
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Nefopam Tricyclic antidepressants (e.g., amitriptyline#) Nav1.7/1.8-selective: DSP-2230§
Funapide§ PF-05089771§
Suzetrigine Pot****ium
openers Flupirtine‡...
-
Nefopam Tricyclic antidepressants (e.g., amitriptyline#) Nav1.7/1.8-selective: DSP-2230§
Funapide§ PF-05089771§
Suzetrigine Pot****ium
openers Flupirtine‡...
-
Nefopam Tricyclic antidepressants (e.g., amitriptyline#) Nav1.7/1.8-selective: DSP-2230§
Funapide§ PF-05089771§
Suzetrigine Pot****ium
openers Flupirtine‡...
-
Nefopam Tricyclic antidepressants (e.g., amitriptyline#) Nav1.7/1.8-selective: DSP-2230§
Funapide§ PF-05089771§
Suzetrigine Pot****ium
openers Flupirtine‡...
-
Proxymetacaine Risocaine Tetracaine Trimecaine Analgesics: AZD-3161 DSP-2230
Funapide GDC-0276 NKTR-171 PF-04531083 PF-05089771
Ralfinamide Raxatrigine RG7893...
-
Nefopam Tricyclic antidepressants (e.g., amitriptyline#) Nav1.7/1.8-selective: DSP-2230§
Funapide§ PF-05089771§
Suzetrigine Pot****ium
openers Flupirtine‡...
-
Proxymetacaine Risocaine Tetracaine Trimecaine Analgesics: AZD-3161 DSP-2230
Funapide GDC-0276 NKTR-171 PF-04531083 PF-05089771
Ralfinamide Raxatrigine RG7893...