-
either an
autoreceptor or a heteroreceptor,
depending upon the type of
transmitter released by the cell on
which it is embedded.
Autoreceptors may be located...
-
while SRAs will
initially byp****
autoreceptors, the
increase in
serotonin they
induce will then
agonise autoreceptors.] In
contrast to SRAs,
SSRIs may...
-
autoreceptors,
which negatively regulate the
release of histamine. The drug
enhances the
activity of
histaminergic neurons by
blocking autoreceptors,...
-
agonist of both
presynaptic 5-HT1A receptors,
which are
inhibitory autoreceptors, and
postsynaptic 5-HT1A receptors. It is
thought that the main effects...
-
presynaptic autoreceptors (low dose) and
postsynaptic D2
receptors (at
higher doses)
antagonist D2sh
selective (presynaptic
autoreceptors) Amisulpride...
-
mediated by
functional selectivity and/or
preferentially binding to D2
autoreceptors at low doses,
resulting in
increased postsynaptic activation via higher...
- 1986). "Identity of
inhibitory presynaptic 5-hydroxytryptamine (5-HT)
autoreceptors in the rat
brain cortex with 5-HT1B
binding sites". Naunyn-Schmiedeberg's...
- of
presynaptic α2
autoreceptors in the CNS
which suppress sympathetic outflow.
Mirtazapine itself blocks these same α2
autoreceptors, so the
effect of...
- 5-HT3, 5-HT6, and/or 5-HT7 in some cases. By
blocking α2-adrenergic
autoreceptors and heteroreceptors, N****As
enhance adrenergic and
serotonergic neurotransmission...
- the
release of
dopamine in the
prefrontal cortex,
through inhibiting autoreceptors.
Further complicating things is the
efficacy of amphetamines, decreased...
