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Lorglumide (CR-1409) is a drug
which inhibits gastrointestinal motility and
reduces gastric secretions,
acting as a
cholecystokinin antagonist, with fairly...
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lorcaserin (USAN) Lorcet-HD
lorcinadol (INN)
loreclezole (INN)
Lorelco Lorfan lorglumide (INN)
lormetazepam (INN)
lornoxicam (INN)
lorpiprazole (INN)
Lorstat Lortab...
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gastric secretions, and
despite older selective CCKA
antagonists such as
lorglumide and
devazepide having had only
limited success in
trials and ultimately...
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other of the CCK receptors.
Selective CCKA
receptor antagonists such as
lorglumide and
devazepide have been
developed both for
their anti-ulcer
effects and...
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Lavigne GJ,
Quirion R (May 1990). "Cholecystokinin
antagonists proglumide,
lorglumide and benzotript, but not L-364,718,
interact with
brain opioid binding...
- Antagonists:
Amiglumide Asperlicin Devazepide Dexloxiglumide Lintitript Lorglumide Loxiglumide Pranazepide Proglumide Tarazepide Tomoglumide Agonists: Cholecystokinin...
- IC50 3.7nM, 1200x
selectivity over CCKB, CAS# 130408-77-4
Proglumide Lorglumide Devazepide Dexloxiglumide Asperlicin SR-27897 IQM-95333 JNJ-17156516 Cholecystokinin...
-
Antagonists Amiglumide Asperlicin Devazepide Dexloxiglumide Lintitript Lorglumide Loxiglumide Pranazepide Proglumide Tarazepide Tomoglumide Agonists Cholecystokinin...
