- are known, 2-
imidazolines, 3-
imidazolines, and 4-
imidazolines. The 2- and 3-
imidazolines contain an
imine center,
whereas the 4-
imidazolines contain an...
-
Imidazoline receptors are the
primary receptors on
which clonidine and
other imidazolines act.
There are
three main
classes of
imidazoline receptor: I1...
-
peripheral vasomotor structures.
Rilmenidine shows greater selectivity for
imidazoline receptors than for
cerebral alpha2-adrenergic receptors, distinguishing...
- 2-
Imidazoline (Preferred
IUPAC name: 4,5-dihydro-1H-imidazole) is one of
three isomers of the nitrogen-containing
heterocycle imidazoline, with the formula...
-
Moxonidine (INN) is a new-generation alpha-2/
imidazoline receptor agonist antihypertensive drug
licensed for the
treatment of mild to
moderate essential...
-
example of autoreceptor. However, it is now
known that
clonidine binds to
imidazoline receptors with a much
greater affinity than α2 receptors,
which would...
- symptoms).
Selected examples are:
Clonidine (mixed alpha2-adrenergic and
imidazoline-I1
receptor agonist)
Dexmedetomidine Fadolmidine Guanfacine, (preference...
- targets:
Neurotransmitter receptors and
receptor ionop****s. Nicotinic,
imidazoline I1 and I2, α2-adrenergic,
glutamate NMDAr, and
serotonin 5-HT2A and 5HT-3...
-
ingested the drug.
There is no
antidote for
tetryzoline or
other similar imidazoline analogue poisoning, but the
symptoms can be alleviated. With treatment...
-
selective α2
adrenergic receptor antagonist, and an
antagonist for the
imidazoline receptor.
Idazoxan has been
under investigation as an antidepressant...
