-
EPPTB, also
known as RO5212773 or RO-5212773, is a drug
developed by Hoffmann-La
Roche which acts as a
potent and
selective antagonist or
inverse agonist...
- RO5256390, the TAAR1
partial agonist RO5263397, and the TAAR1
antagonists EPPTB and RTI-7470-44.
Selective TAAR1
agonists are used in
scientific research...
- is
reduced by the
trace amine-****ociated
receptor 1 (TAAR1)
antagonist EPPTB. In addition, the HTR of 5-HTP is
abolished by
indolethylamine N-methyltransferase...
- the
trace amine-****ociated
receptor 1 (TAAR1).
Antagonists of MAEs, like
EPPTB (a
known TAAR1 antagonist), 3-F-BPAP, and rasagiline, have been identified...
- TAAR1 to be identified,
following the
potent mouse TAAR1
inverse agonist EPPTB in 2009. The
affinity (Ki) of RTI-7470-44 for the
human TAAR1 is 0.3 nM...
-
effects were
absent with TAAR1
knockout mice or with the TAAR1
antagonist EPPTB. In addition, T1AM-mediated TH
phosphorylation appeared to be
mediated by...
-
Agonists Antagonists Compound 22
EPPTB (RO-5212773) RTI-7470-44
Inverse agonists EPPTB (RO-5212773)...
-
Agonists Antagonists Compound 22
EPPTB (RO-5212773) RTI-7470-44
Inverse agonists EPPTB (RO-5212773)...
-
Agonists Antagonists Compound 22
EPPTB (RO-5212773) RTI-7470-44
Inverse agonists EPPTB (RO-5212773)...
-
Agonists Antagonists Compound 22
EPPTB (RO-5212773) RTI-7470-44
Inverse agonists EPPTB (RO-5212773)...
