-
Benzomorphan is a
chemical compound that is the base for a
series of
drugs which variably act on the
opioid kappa and
sigma receptors,
including the following...
-
Ketazocine (INN), also
known as ketocyclazocine, is a
benzomorphan derivative used in
opioid receptor research. Ketazocine, for
which the
receptor is named...
-
Benzomorphans 8-CAC
Alazocine Bremazocine Dezocine Ketazocine Metazocine Pentazocine Phenazocine Cyclazocine 4-Phenylpiperidines 4-Fluoromeperidine Allylnorpethidine...
- a much more
potent analgesic than
pentazocine and
other drugs in the
benzomorphan series, most
probably due to the
presence of an N-phenethyl substitution...
- ATC code N02
Analgesics is a
therapeutic subgroup of the
Anatomical Therapeutic Chemical classification System, a
system of
alphanumeric codes developed...
- in most
countries in the same
fashion as is morphine. The
prototype benzomorphan,
metazocine (6), can be
obtained from a
variation of the
morphinan synthesis...
-
pentazocine and phenazocine. This
family of
opioid drugs is
called the
benzomorphans or benzazocines. It is a KOR
agonist and MOR
partial agonist, and also...
-
obtained by
increasing the dose any further.
Chemically it is
classed as a
benzomorphan and it
comes in two enantiomers,
which are
molecules that are exact...
- As per codeine.
Respiratory depression is
subject to
ceiling effect.
Benzomorphans Dezocine No data available.
Mixed opioid agonist-antagonist. IM, IV...
- breathing. The
crystal structure of
bremazocine was
determined in 1984
Benzomorphan Dortch-Carnes J,
Potter DE (2005). "Bremazocine: a kappa-opioid agonist...
